Bisoprololum Index Natura Bisoprololi | Notae | Nexus interniTabula navigationisWHO"Pharmacokinetics and metabolism of bisoprolol enantiomers in humans"

Ordinis mundi sanitarii medicamenta principaliaAntiarrhythmica


antiarrhythmicumordinis mundi sanitariiindicem exemplarem medicamentorum principaliumbeta1-receptoriorumRSCodex ATCC07AB07Tempus semivitae biologicumCytochromatis P450 CYP2D6CYP3A4CYP3A4







Esculaap4.svg


Cave: notitiae huius paginae nec praescriptiones nec consilia medica sunt.


Bisoprololum est substantia chemica beta-receptoria typi primi inhibens et propterea medicamentum antihypertensivum velut antiarrhythmicum classis II est.


Bisoprololum in ordinis mundi sanitarii indicem exemplarem medicamentorum principalium receptum est.




Index





  • 1 Natura Bisoprololi

    • 1.1 Natura chemica


    • 1.2 Natura pharmacologica


    • 1.3 Pharmacocinetica


    • 1.4 Interactiones



  • 2 Notae


  • 3 Nexus interni




Natura Bisoprololi |



Natura chemica |





Bisoprololum beta1-receptoria valde selective inhibet.


Bisoprololum est beta1-receptoriorum inhibitor. Structura eius chemica est (RS)-1-[4-(2-isopropoxyethoxymethyl)phenoxy]-3-isopropylamino-2-propanolum.


Formula chemica est C18H31NO4, massa molaris 325.45 g/mol.
Codex ATC est C07AB07 (WHO).



Natura pharmacologica |



Pharmacocinetica |


Solubilitas in aqua est 2.24 g·mol−1 (25 °C), accessibilitas biologica 90%.
Tempus semivitae biologicum t12displaystyle t_frac 12.[1]10 – 12 h est.


Bisoprololum substratum et Cytochromatis P450 CYP2D6 ( (R)-(+)-bisoprololum > (S)-(-)-bisoprololum ) et CYP3A4 ( (R)=(S) ) est.[2]



Interactiones |


Cum Bisoprololum subtratum enzymi CYP3A4 esset, inhibitores CYP3A4 effectus Bisoprololi augere possint, inductores invicem diminuere, per exemplum:







Pharmaca cum effectibus Bisoprololi substrati
Inhibitores cum Bisoprololi effectibus fortioribus
Inductores cum Bisoprololi effectibus minoribus

  • Antihypertensiva

    • Calcii canalium inhibitores
      • Diltiazemum

      • Felodipinum



  • Antiarrhythmica
    • Amiodaronum

  • Diuretica/Hormonta

    • Conivaptanum (forte)


  • Antibiotica
    • Ciprofloxacinum


    • Clarithromycinum (forte)


    • Erythromycinum (forte)


    • Telithromycinum (forte)


  • Fungicida/-statica

    • Ketoconazolum (forte)


    • Itraconazolum (forte)


    • Posaconazolum (forte)


    • Voriconazolum (forte)


  • Proteasis inhibitores
    • Atazanavirum-Ritonavirum


    • Boceprevirum (forte)


    • Ritonavirum (forte)


    • Indinavirum (forte)


    • Nelfinavirum (forte)


    • Saquinavirum (forte)


    • Telaprevirum (forte)


  • Antidepressiva

    • Nefazodonum (forte)

  • Glucocorticoides

    • Dexamethasonum (forte)


  • Hormonta
    • GH


  • Plantae
    • Fructus averrhoae carambolae

    • Silybum marianum



  • Anticonvulsiva

    • Carbamazepinum (forte, quoque P-gp)


    • Phenytoinum (forte)


    • Fosphenytoinum (forte)


    • Oxcarbazepinum (forte)

    • Topiramatum


    • Phenobarbitalum (forte)


    • Primidonum (forte)


  • Antidepressiva

    • Hypericum perforatum (forte, quoque P-gp)

  • Antihypertensiva

    • Bosentanum (forte, endothelini receptoris inhibitor)

  • Substantiae antiretrovirales

    • Efavirenzum (forte)


    • Etravirinum (forte)


    • Nevirapinum (forte)


  • Substantiae antineoplasticae
    • Enzalutamidum


    • Mitotanum (forte)



  • Antibiotica

    • Rifabutinum (forte)


    • Rifapentinum (forte)


    • Nafcillinum (forte)


    • Rifampicinum (forte)



  • Hormonta
    • Triiodthyroninum (T3)

  • Modafinilum

  • Quercetinum

  • Capsaicinum


Notae |



  1. ↑ http://goldbook.iupac.org/B00658.html


  2. ↑ Yuji Horikiri; Takehiko Suzuki; Masakazu Mizobe (March 1998). "Pharmacokinetics and metabolism of bisoprolol enantiomers in humans". Journal of Pharmaceutical Sciences 87 (3): 289–294 


Nexus interni


  • Cor

-

Popular posts from this blog

strTok function (thread safe, supports empty tokens, doesn't change string)String case reverse function in CGet line from string functionTDD: String Calculator KataC - K&R getint() variationSimple function to generate an HTML-safe stringGeneric Pairing Heap PerformancePattern for writing a generic string transformation functionChange a string into a function/def activatorC++ string tokenizing without streams, with certain conditionsRead consecutive blanks in array

Image
What are these boxed doors outside store fronts in New York? RSA: Danger of using p to create q Theorems that impeded progress strTok function (thread safe, supports empty tokens, doesn't change string) What typically incentivizes a professor to change jobs to a lower ranking university? Accidentally leaked the solution to an assignment, what to do now? (I'm the prof) I'm flying to France today and my passport expires in less than 2 months Watching something be written to a file live with tail Alternative to sending password over mail? Today is the Center Why "Having chlorophyll without photosynthesis is actually very dangerous" and "like living with a bomb"? Languages that we cannot (dis)prove to be Context-Free Did Shadowfax go to Valinor? How is it possible to have an ability score that is less than 3? Is it tax fraud for an individual to declare non-taxable revenue as taxable income? (US tax laws) Why is 150k or 200k job...
Read more

How to write “ä” and other umlauts and accented letters in bibliography?Accents in BibTeXSorting references with special characters alphabeticallyUse ae ligature in bibliographyEastern European nameInverted circumflex in BibTexBibTex, non-ascii initials and nameptr fproblems with accent in LatexHow to add a Ø to my bibliography from Jabref?References without accentsTroubles when trying to cite St“omer-Verlet in ”title" field of a bib entryComprehensive list of accented charactersHow to type the letter “i” with two dots (diaeresis) in math mode?Problem with glossary text and accented lettersSpecial character in bibliographyAccented letters, Unicode and LaTeX accentsHow to stop natbib from modifying bibliography styleCitation of a paper with non-standard characters by BibtexWrite accented characters to file using writeHow to group the bibliography alphabetically, if some surnames start with “accented” characters?How can I automatically capitalize significant words in my bibliography?

Image
Information to fellow intern about Hiring? Are tax years 2016 & 2017 back taxes deductible for tax year 2018? Why a const reference doesn't extend the life of temporary object passed via function? Why did the Germans forbid the possession of pet pigeons in Rostov-on-Don in 1941? I see my dog run How to avoid repetitive long generic constraints in Rust How can I fix this gap between bookcases I made? What are these boxed doors outside store fronts in New York? How would photo IDs work for shapeshifters? What does "enim et" mean? What is the meaning of "of trouble" in the following sentence? How to determine if window is maximised or minimised from bash script Calculate Levenshtein distance between two strings in Python Why do we use polarized capacitors? How to answer pointed "are you quitting" questioning when I don't want them to suspect Extreme, but not acceptable situation and I can't start the work tomorrow...
Read more

Title of papers that have not been submitted to a venue?How “submitted”, “to appear”, “accepted” papers are evaluated in a CV?What percentage of papers submitted to a conference or journal have been previously rejected in the same or another venue?How to automatically extract submitted/accepted dates of many journal papers?Is it okay/common/good to mention the submitted papers in my phd thesis?Can one determine whether somebody's work may have been plagiarized?How to describe a paper for which you have not yet submitted revisions in CV?JCR publication required to enrol in PhD program - is it common?“Full” versions versus “Preliminary” version of result/paper. Are they considered different?How can I prove that my article has not been submitted to another journal?Is there anything that has been tried to stop publication shopping

Image
Can I write a for loop that iterates over both collections and arrays? Is it possible for the two major parties in the UK to form a coalition with each other instead of a much smaller party? What is the command to reset a Windows installation without deleting any files How to answer pointed "are you quitting" questioning when I don't want them to suspect Can I legally use front facing blue light in the UK? Is "plugging out" electronic devices an American expression? Why is the design of haulage companies so “special”? What is the steepest angle that a canal can be traversable without locks? Patience, young "Padovan" Is this food a bread or a loaf? Geography at the pixel level Symbol above others Springs with some finite mass Why do UK politicians seemingly ignore opinion polls on Brexit? Is there a name of the flying bionic bird? What does 'script /dev/null' do? Is std::next for vector O(n) or O(1)? Are cabin d...
Read more